Search Result "dual-site binding"


Peripheral and Dual Binding Site Acetylcholinesterase Inhibitors: Implications in treatment of Alzheimers Disease

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 1 Issue: 3 Year: 2001 Page: 267-272
Author(s): Ana Castro, Ana Martinez

Structural Determinants of the Multifunctional Profile of Dual Binding Site Acetylcholinesterase Inhibitors as Anti-Alzheimer Agents

Journal: Current Pharmaceutical Design
Volume: 16 Issue: 2 Year: 2010 Page: 2818-2836
Author(s): Carles Galdeano, Elisabet Viayna, Pau Arroyo, Axel Bidon-Chanal, J. Ramon Blas, Diego Munoz-Torrero, F. Javier Luque

From Dual Binding Site Acetylcholinesterase Inhibitors to Multi-Target-Directed Ligands (MTDLs): A Step Forward in the Treatment of Alzheimers Disease

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2008 Page: 960-967
Author(s): Maria Laura Bolognesi, Anna Minarini, Michela Rosini, Vincenzo Tumiatti, Carlo Melchiorre

Design and Synthesis of New Dual Binding Site Cholinesterase Inhibitors: in vitro Inhibition Studies with in silico Docking

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 3 Year: 2014 Page: 331-338
Author(s): Muhammad Yar,Marek Bajda,Rana Atif Mehmood,Lala Rukh Sidra,Nisar Ullah,Lubna Shahzadi,Muhammad Ashraf,Tayaba Ismail,Sohail Anjum Shahzad,Zulfiqar Ali Khan,Syed Ali Raza Naqvi,Nasir Mahmood

Review Article

Specificity of Binding in Protein Kinases

Journal: Current Enzyme Inhibition
Volume: 13 Issue: 2 Year: 2017 Page: 89-98
Author(s): Satya P. Gupta, Basheerulla Shaik, Vijay K. Agrawal

Fetzima (levomilnacipran), a Drug for Major Depressive Disorder as a Dual Inhibitor for Human Serotonin Transporters and Beta-Site Amyloid Precursor Protein Cleaving Enzyme-1

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 13 Issue: 8 Year: 2014 Page: 1427-1431
Author(s): Syed Mohd. Danish Rizvi,Sibhghatulla Shaikh,Mahiuddin Khan,Deboshree Biswas,Nida Hameed,Shazi Shakil

The Role of Binding Kinetics in GPCR Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 15 Issue: 24 Year: 2015 Page: 2504-2522
Author(s): David C. Swinney,Brad A. Haubrich,Isabelle Van Liefde,Georges Vauquelin

Targeting Beta-Amyloid Pathogenesis Through Acetylcholinesterase Inhibitors

Journal: Current Pharmaceutical Design
Volume: 12 Issue: 3 Year: 2006 Page: 4377-4387
Author(s): Ana Castro, Ana Martinez

Structural Insight into PPARγ Ligands Binding

Journal: Current Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2009 Page: 1768-1789
Author(s): A. Farce, N. Renault, P. Chavatte

Structural Identification of DnaK Binding Sites within Bovine and Sheep Bactenecin Bac7

Journal: Protein & Peptide Letters
Volume: 21 Issue: 4 Year: 2014 Page: 407-412
Author(s): Michael Zahn,Bjorn Kieslich,Nicole Berthold,Daniel Knappe,Ralf Hoffmann,Norbert Strater

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